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| | Morphothiadin Basic information |
| Product Name: | Morphothiadin | | Synonyms: | Morphothiadin;GLS4
(GLS 4;5-Pyrimidinecarboxylic acid, 4-(2-bromo-4-fluorophenyl)-1,4-dihydro-6-(4-morpholinylmethyl)-2-(2-thiazolyl)-, ethyl ester;Morphothiadin USP/EP/BP;GLS 4(Morphothiadin);Morphothiadin (GLS4);Morphothiadin,inhibit,HBV,Inhibitor,GLS-4,GLS 4,Hepatitis B virus | | CAS: | 1092970-12-1 | | MF: | C21H22BrFN4O3S | | MW: | 509.39 | | EINECS: | | | Product Categories: | | | Mol File: | 1092970-12-1.mol |  |
| | Morphothiadin Chemical Properties |
| Boiling point | 577.2±60.0 °C(Predicted) | | density | 1.58±0.1 g/cm3(Predicted) | | storage temp. | Store at -20°C | | solubility | DMF: 12 mg/ml; DMSO: 1 mg/ml; Ethanol: Slightly soluble; PBS (pH 7.2): 0.3 mg/ml | | form | A solid | | pka | 8.38±0.10(Predicted) |
| | Morphothiadin Usage And Synthesis |
| Uses | Morphothiadin, is a potent inhibitor on the replication of both wild-type and adefovir-resistant HBV with an IC50 of 12 nM. It strongly inhibits virus accumulation in the supernatant of HepAD38 cells at 25 nM to 100 nM (P<0.02). |
| | Morphothiadin Preparation Products And Raw materials |
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