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| | Cefetrizole Basic information |
| Product Name: | Cefetrizole | | Synonyms: | Cefetrizole;(6R,7R)-8-Oxo-7-[2-thienylacetylamino]-3-[(1H-s-triazol-3-ylthio)methyl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid;5-Thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid, 8-oxo-7-[[2-(2-thienyl)acetyl]amino]-3-[(1H-1,2,4-triazol-5-ylthio)methyl]-, (6R,7R)- | | CAS: | 65307-12-2 | | MF: | C16H15N5O4S3 | | MW: | 437.52 | | EINECS: | | | Product Categories: | | | Mol File: | 65307-12-2.mol |  |
| | Cefetrizole Chemical Properties |
| density | 1.71±0.1 g/cm3(Predicted) | | pka | 2.65±0.50(Predicted) |
| | Cefetrizole Usage And Synthesis |
| Biological Activity | Ceftezole is an α-Glucosidase inhibitor with IC50 and Ki values of 2.1 μM and 0.578 μM, respectively. | | in vitro | In in vitro α-Glucosidase assays, Ceftezole is shown to be a reversible, non-competitive inhibitor of yeast α-glucosidase with a K i value of 5.78×10 -7 M when the enzyme mixture is pretreated with ceftezole. | | target | IC50: 2.1 μM (α-Glucosidase)
Ki: 0.578 μM (α-Glucosidase) |
| | Cefetrizole Preparation Products And Raw materials |
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